Azamulin
- $45 - $2000
- Product name: Azamulin
- CAS: 76530-44-4
- MF: C24H38N4O4S
- MW: 478.65
- EINECS:
- MDL Number:MFCD00865055
- Synonyms:SA 85530b;14-O-(5-(2-Amino1,3,4-triazolyl)thioacetyl)dihydromutilin;Antibiotic TDM 85-530;Azamulin;[(5-Amino-1H-1,2,4-triazol-3-yl)thio]acetic acid (3aS,4R,5S,6R,8R,9R,9aR,10R)-6-ethyldecahydro-5-hydroxy-4,6,9,10-tetramethyl-1-oxo-3a,9-propano-3aH-cyclopentacycloocten-8-yl ester;TMD 85-530, SA 85530b;Acetic acid, 2-[(3-amino-1H-1,2,4-triazol-5-yl)thio]-, (3aS,4R,5S,6R,8R,9R,9aR,10R)-6-ethyldecahydro-5-hydroxy-4,6,9,10-tetramethyl-1-oxo-3a,9-propano-3aH-cyclopentacycloocten-8-yl ester
9 prices
Selected condition:
Brand
- AK Scientific
- Cayman Chemical
- Medical Isotopes, Inc.
- Sigma-Aldrich
- TRC
Package
- 500μg
- 1mg
- 2mg
- 5mg
- 25mg
- ManufacturerAK Scientific
- Product number6562BB
- Product descriptionAzamulin
- Packaging1mg
- Price$199
- Updated2021-12-16
- Buy
- ManufacturerCayman Chemical
- Product number18748
- Product descriptionAzamulin ≥98%
- Packaging500μg
- Price$45
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number18748
- Product descriptionAzamulin ≥98%
- Packaging1mg
- Price$73
- Updated2024-03-01
- Buy
- ManufacturerCayman Chemical
- Product number18748
- Product descriptionAzamulin ≥98%
- Packaging5mg
- Price$180
- Updated2024-03-01
- Buy
- ManufacturerMedical Isotopes, Inc.
- Product number6969
- Product descriptionAzamulin
- Packaging5mg
- Price$875
- Updated2021-12-16
- Buy
- ManufacturerMedical Isotopes, Inc.
- Product number6969
- Product descriptionAzamulin
- Packaging25mg
- Price$2000
- Updated2021-12-16
- Buy
- ManufacturerSigma-Aldrich
- Product numberSML0485
- Product descriptionAzamulin ≥98% (HPLC)
- Packaging5mg
- Price$201
- Updated2024-03-01
- Buy
- ManufacturerSigma-Aldrich
- Product numberSML0485
- Product descriptionAzamulin ≥98% (HPLC)
- Packaging25mg
- Price$774
- Updated2024-03-01
- Buy
- ManufacturerTRC
- Product numberA801530
- Product descriptionAzamulin
- Packaging2mg
- Price$110
- Updated2021-12-16
- Buy
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|
AK Scientific | 6562BB | Azamulin | 1mg | $199 | 2021-12-16 | Buy |
Cayman Chemical | 18748 | Azamulin ≥98% | 500μg | $45 | 2024-03-01 | Buy |
Cayman Chemical | 18748 | Azamulin ≥98% | 1mg | $73 | 2024-03-01 | Buy |
Cayman Chemical | 18748 | Azamulin ≥98% | 5mg | $180 | 2024-03-01 | Buy |
Medical Isotopes, Inc. | 6969 | Azamulin | 5mg | $875 | 2021-12-16 | Buy |
Medical Isotopes, Inc. | 6969 | Azamulin | 25mg | $2000 | 2021-12-16 | Buy |
Sigma-Aldrich | SML0485 | Azamulin ≥98% (HPLC) | 5mg | $201 | 2024-03-01 | Buy |
Sigma-Aldrich | SML0485 | Azamulin ≥98% (HPLC) | 25mg | $774 | 2024-03-01 | Buy |
TRC | A801530 | Azamulin | 2mg | $110 | 2021-12-16 | Buy |
Properties
Melting point :128-130°C
Boiling point :659.4±65.0 °C(Predicted)
Density :1.27±0.1 g/cm3(Predicted)
storage temp. :-20°C
solubility :DMSO: soluble10mg/mL (clear solution)
form :powder
pka :9.56±0.40(Predicted)
color :white to beige
Stability :Store at -2℃.
Boiling point :659.4±65.0 °C(Predicted)
Density :1.27±0.1 g/cm3(Predicted)
storage temp. :-20°C
solubility :DMSO: soluble10mg/mL (clear solution)
form :powder
pka :9.56±0.40(Predicted)
color :white to beige
Stability :Store at -2℃.
Safety Information
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Signal word: | Warning | ||||||||||||||||||||||||||||
Hazard statements: |
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Precautionary statements: |
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Description
Azamulin is a selective, irreversible inhibitor of cytochrome P450 (CYP) 3A isoforms (IC50 values range from 26 to 240 nM for CYP3A4 and CYP3A4/5 from different sources). It is at least 50-fold less potent against CYP2J2 and 100-fold less effective against all other CYP isoforms. Azamulin potently blocks the hydroxylation of testosterone and midazolam by CYP3A4.Related product price
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$110