生物活性
Lasmiditan succinate (COL-144, LY573144)是一種新型的、作用于中樞神經(jīng)系統(tǒng)的5-HT(1F) receptor激動劑,Ki值為2.21 nM,無收縮血管活性。
英文同義詞
2,4,6-trifluoro-N-{6-[(1-methylpiperidine-4-yl)carbonyl]pyridin-2-yl}benzamidehemisuccinate;LASMIDITANSUCCINATE;Lasmiditanhemisuccinate;Lasmiditansuccinate(USAN);2,4,6-Trifluoro-N-[6-[(1-methyl-4-piperidinyl)carbonyl]-2-pyridinyl]benzamide,butanedioicacid(1:2);Lasmiditansuccinate(Synonyms:COL-144succinate;LY573144succinate);butanedioicacid,compd.with2,4,6-trifluoro-n-(6-((1-methyl-4-piperidinyl)carbonyl)-2-pyridinyl)benzamide
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