Description: |
Selective urotensin-II (UT) receptor antagonist (Ki values are 61, 17, 30, 65 and 56 nM at human, monkey, cat, rat and mouse receptors respectively). Inhibits U-II-induced intracellular Ca2+mobilization (IC50 = 180 nM) and antagonizes the contractile action of U-II in isolated mammalian arteries and aortae (EC50 = 50 - 189 nM).For the detailed information of SB-657510, the solubility of SB-657510 in water, the solubility of SB-657510 in DMSO, the solubility of SB-657510 in PBS buffer, the animal experiment (test) of SB-657510, the cell expriment (test) of SB-657510, the in vivo, in vitro and clinical trial test of SB-657510, the EC50, IC50,and Affinity of SB-657510, Please contact DC Chemicals. |