Tenidap NEW
| Price | $30 | $64 | $109 |
| Package | 1mg | 5mg | 10mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2024-11-14 |
Product Details
| Product Name: Tenidap | CAS No.: 120210-48-2 |
| Purity: 99.42% | Supply Ability: 10g |
| Release date: 2024/11/14 |
Product Introduction
Bioactivity
| 名稱 | Tenidap |
| 描述 | Tenidap (CP-66248) is a selective COX-1 and SLC26A3 inhibitor with anti-inflammatory, analgesic, and anti-rheumatic activities. |
| 體外活性 | The human astrocytoma cell line U373 MG was incubated with 0.1-100 μM tenidap for 30 min and then stimulated with 50 μM C6-ceramide for 24 h. Tenidap inhibited the dose-dependent ceramide-induced IL-6 protein synthesis in U373 human astrocytoma cells.[4] |
| 體內(nèi)活性 | After sustained epilepsy (SE) induced by trichostatin in male Wistar rats, Tenidap was administered at 10 mg / kg daily for 10 days, 46.88 ± 10.70 neurons survived in the tenidap-SE group, and 37.75 ± 8.78 neurons survived in the tenidap-SE group, Tenidap significantly inhibited the hippocampal expression of COX-2 in the hippocampus, especially in the CA3 region.[3] |
| 存儲(chǔ)條件 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| 溶解度 | DMSO : 20 mg/mL (62.35 mM), Sonication is recommended. |
| 關(guān)鍵字 | Tenidap | CP66248 | CP 66248 |
| 相關(guān)產(chǎn)品 | 5-Fluorouracil | Bismuth Subsalicylate | Procaine | Ibuprofen | Acetaminophen | Guanidine hydrochloride | Diclofenac sodium | Diclofenac Potassium | N-Nitrosodiethylamine | Thymidine | Paradol | Salicylic acid |
| 相關(guān)庫 | 抗結(jié)直腸癌化合物庫 | 非甾體類抗炎化合物庫 | DNA 損傷和修復(fù)分子庫 | 疼痛相關(guān)化合物庫 | 經(jīng)典已知活性庫 | HIF-1化合物庫 | 抗乳腺癌化合物庫 | 抑制劑庫 | 抗衰老化合物庫 | 免疫/炎癥分子化合物庫 | 已知活性化合物庫 | 人代謝物化合物庫 |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
You may like
Recommended supplier
| Product name | Price | Suppliers | Update time | |
|---|---|---|---|---|
| $1670.00/25mg |
VIP1Y
|
TargetMol Chemicals Inc.
|
2024-10-28 | |
| $1.10/1g |
VIP4Y
|
Dideu Industries Group Limited
|
2021-07-06 | |
| $1.10/1g |
VIP4Y
|
Dideu Industries Group Limited
|
2021-07-06 |
United States- Since: 2011-01-07
- Address: 36?Washington?Street, Wellesley?Hills
INQUIRY