224579-74-2
中文名稱
MYOSIN LIGHT CHAIN KINASE INHIBITOR PEPTIDE 18
英文名稱
MLCK INHIBITOR PEPTIDE 18
CAS
224579-74-2
分子式
C60H105N23O11
分子量
1324.62
MOL 文件
224579-74-2.mol
更新日期
2024/10/20 11:23:30
224579-74-2 結(jié)構(gòu)式
基本信息
中文別名
MLCK抑制肽18MLCK抑制肽18?, >98%
英文別名
H-RKKYKYRRK-NH2MLCK INHIBITOR PEPTIDE 18
MLCK inhibitor peptide 18,RKKYKYRRK, >98%
MYOSIN LIGHT CHAIN KINASE INHIBITOR PEPTIDE 18
L-Lysinamide, L-arginyl-L-lysyl-L-lysyl-L-tyrosyl-L-lysyl-L-tyrosyl-L-arginyl-L-arginyl-
物理化學(xué)性質(zhì)
密度1.44±0.1 g/cm3(Predicted)
儲(chǔ)存條件Desiccate at -20°C
溶解度DMF: 12 mg/mL; DMSO: 5 mg/mL; Ethanol: 12 mg/mL; PBS (pH 7.2): 5 mg/mL
酸度系數(shù)(pKa)9.82±0.15(Predicted)
形態(tài)結(jié)晶固體
顏色White to off-white
水溶解性Soluble to 1 mg/ml in water
序列H-Arg-Lys-Lys-Tyr-Lys-Tyr-Arg-Arg-Lys-NH2
MYOSIN LIGHT CHAIN KINASE INHIBITOR PEPTIDE 18價(jià)格(試劑級(jí))
| 報(bào)價(jià)日期 | 產(chǎn)品編號(hào) | 產(chǎn)品名稱 | CAS號(hào) | 包裝 | 價(jià)格 |
| 2024/08/19 | HY-P1029 | MYOSIN LIGHT CHAIN KINASE INHIBITOR PEPTIDE 18 MLCK inhibitor peptide 18 | 224579-74-2 | 1mg | 500元 |
| 2024/08/19 | HY-P1029 | MYOSIN LIGHT CHAIN KINASE INHIBITOR PEPTIDE 18 MLCK inhibitor peptide 18 | 224579-74-2 | 5mg | 1750元 |
| 2024/08/19 | HY-P1029 | MYOSIN LIGHT CHAIN KINASE INHIBITOR PEPTIDE 18 MLCK inhibitor peptide 18 | 224579-74-2 | 10mg | 3200元 |
常見問題列表
生物活性
MLCK inhibitor peptide 18 是一種有效的 MLCK 抑制劑，IC50 值為 50 nM，同時(shí)較弱抑制 CaM kinase II 的活性。靶點(diǎn)
IC50: 50 nM (MLCK)
體外研究
MLCK inhibitor peptide 18 has a selective effect on peptide substrate utilization by MLCK, does not interfere with kinase activation by CaM, does not have significant inhibitory activity with the closely related CaMPKII, and does not inhibit PKA.