Identification | Back Directory | [Name]
CINITAPRIDE HYDROGEN TARTRATE | [CAS]
66564-14-5 | [Synonyms]
Cidine LAS-17177 CinitaprideTartrate CINITAPRIDE HYDROGEN TARTRATE 4-Amino-N-[1-(3-cyclohexen-1-ylmethyl)-4-piperidyl]-2-ethoxy-5-nitrobenzamide 4-Amino-N-[1-(3-cyclohexen-1-ylmethyl)-4-piperidinyl]-2-ethoxy-5-nitrobenzamide 4-amino-N-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-2-ethoxy-5-nitrobenzamide BenzaMide,4-aMino-N-[1-(3-cyclohexen-1-ylMethyl)-4-piperidinyl]-2-ethoxy-5-nitro- | [Molecular Formula]
C25H36N4O10 | [MDL Number]
MFCD00897211 | [MOL File]
66564-14-5.mol | [Molecular Weight]
552.57 |
Chemical Properties | Back Directory | [Melting point ]
>197°C (dec.) | [Boiling point ]
579.8±50.0 °C(Predicted) | [density ]
1.24 | [storage temp. ]
Refrigerator | [solubility ]
DMSO (Slightly), Methanol (Slightly), Water (Slightly) | [form ]
Solid | [pka]
12.62±0.20(Predicted) | [color ]
Yellow |
Hazard Information | Back Directory | [Chemical Properties]
White Solid | [Usage]
A novel prokinetic benzamide-stimulating gastrointestinal motility agent and antiucer agent. It acts as an agonist of the 5-HT1 and 5-HT4 receptors and as an antagonist of the 5-HT2 receptors. | [Usage]
serotonin-norepinephrine reuptake inhibitor, antidepressant | [Description]
Cinitapride is a substituted benzamide dopamine receptor antagonist effective in the
treatment of gastroesophageal reflux and a variety of gastrointestinal motility disorders.
It generates strong procholinergic activity in the gastrointestinal tract by elevating the
serotonergic transmission in the mysenteric plexus. | [Originator]
Almirall (Spain) | [Uses]
A novel prokinetic benzamide-stimulating gastrointestinal motility agent and antiucer agent. It acts as an agonist of the 5-HT1 and 5-HT4 receptors and as an antagonist of the 5-HT2 receptors (1,2,3). | [Uses]
A novel prokinetic benzamide-stimulating gastrointestinal motility agent and antiucer agent. It acts as an agonist of the 5-HT1 and 5-HT4 receptors and as an antagonist of the 5-HT2 receptors. | [Uses]
serotonin-norepinephrine reuptake inhibitor, antidepressant | [Definition]
ChEBI: Cinitapride is an aromatic ether and a C-nitro compound. | [Brand name]
Cidine |
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