Identification | Back Directory | [Name]
L 365260 | [CAS]
118101-09-0 | [Synonyms]
260 L-365 L 365260 MSD-365260 L-365260
(L 365260 (3R)-1-Methyl-3-[3-(3-methylphenyl)ureido]-5-phenyl-1H-1,4-benzodiazepin-2(3H)-one 1-[[(3R)-2,3-Dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin]-3-yl]-3-(3-methylphenyl)urea Urea, N-[(3R)-2,3-dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl]-N'-(3-methylphenyl)- (+)-1-[[(3R)-2,3-Dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin]-3-yl]-3-(3-methylphenyl)urea (+)-N-[[(3R)-2,3-Dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin]-3-yl]-N'-(3-methylphenyl)urea | [Molecular Formula]
C24H22N4O2 | [MDL Number]
MFCD00869756 | [MOL File]
118101-09-0.mol | [Molecular Weight]
398.46 |
Hazard Information | Back Directory | [Uses]
L-365,260 is a non-peptide competitive CCK-BR antagonist. | [Definition]
ChEBI: L-365260 is a benzodiazepine. | [Biological Activity]
Selective cholecystokinin receptor 2 (CCK 2 ) antagonist (IC 50 values are 2 and 280 nM at CCK 2 and CCK 1 receptors respectively) that is inactive at a range of other receptors including opiate, muscarinic acetylcholine, α - and β adrenergic, histamine, angiotensin and bradykinin receptors. | [storage]
Store at +4°C |
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